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 药物发现的新方法 872条(本栏目收费,不能显示细节,电话13136136841)
colorectal cancer, 213 213
gemcitabine, 214 214
limitations, 214–215 215
NSCLC model, 213 213
pancreatic cancer, 213–214 214
scope of, 211–213 213
TIV, 204–206 206
TR process, 208–209 209
in vitro screening, 215 215
Predictive biomarkers, 208 208
Privileged structures benzodiazepine scaffold, 113–114 114
combinatorial approach, 115 115
CtB approach, 115 115
quinazolinone privileged scaffold, 114 114
steroid adrenosterone, 115, 116 116
Progesterone receptor antagonists (PRA), 192,194–197 197
Progesterone receptors (PGR), 194–196 196
Proof of concept (PoC), 290 290
Prosigna™ test, 292 292
Prostaglandin H2 (PGH2), 141 141
Protein biomarker, 297 297
Protein databank (PDB), 45 45
Protein–protein interactions (PPIs) 0
in health and disease, 126–127 127
intractable targets 0
acetyl-lysine mimetic inhibitors, 0
bromodomains, 51–52 52
bromodomains, chemical probes,52, 53 53
epigenetic reader domain, 50 50
inhibitors block, 50 50
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