药物发现,开发和制造 499条(本栏目收费,不能显示细节,电话15274084725)
MOLECULAR SIMILARITY
METHODS AND QSAR MODELS AS
TOOLS FOR VIRTUAL SCREENING 87
SYSTEMS BIOLOGY: APPLICATIONS
IN DRUG DISCOVERY 123
HIGH-THROUGHPUT
FLOW CYTOMETRY 185
COMBINING NMR SPECTRAL
INFORMATION WITH ASSOCIATED
STRUCTURAL FEATURES TO
FORM COMPUTATIONALLY
NONINTENSIVE, RUGGED, AND
OBJECTIVE MODELS OF
BIOLOGICAL ACTIVITY 227
USING MICROSOFT EXCEL® AS A
LABORATORY DATA
MANAGEMENT TOOL 287
SIMULTANEOUS SCREENING OF
MULTIPLE CELL LINES USING THE
CELLCARD SYSTEM 353
PROTEIN X-RAY
CRYSTALLOGRAPHY IN
DRUG DISCOVERY 373
BIOLOGICAL AND CHEMISTRY
ASSAYS AVAILABLE DURING
DRUG DISCOVERY AND
DEVELOPABILITY ASSESSMENT 457
STRATEGIES AND METHODS IN
MONITORING AND TARGETING
PROTEIN–PROTEIN INTERACTIONS 483
HIGH-THROUGHPUT SCREENING:
EVOLUTION OF TECHNOLOGY
AND METHODS 559
METAL-ENHANCED
FLUORESCENCE: APPLICATION TO
HIGH-THROUGHPUT SCREENING
AND DRUG DISCOVERY 603
METHODS FOR THE DESIGN
AND ANALYSIS OF
REPLICATE-EXPERIMENT
STUDIES TO ESTABLISH
ASSAY REPRODUCIBILITY
AND THE EQUIVALENCE OF
TWO POTENCY ASSAYS 667
COUPLED LUMINESCENT
METHODS IN DRUG DISCOVERY:
3-MIN ASSAYS FOR CYTOTOXICITY
AND PHOSPHATASE ACTIVITY 689
DESIGN AND PHARMACEUTICAL
APPLICATIONS OF PRODRUGS 733
GABA AND GLUTAMATE
RECEPTOR LIGANDS AND
THEIR THERAPEUTIC
POTENTIAL IN CNS DISORDERS 797
CARDIAC SARCOLEMMAL
ATP-SENSITIVE POTASSIUM
CHANNEL ANTAGONISTS:
NOVEL ISCHEMIA-SELECTIVE
ANTIARRHYTHMIC AGENTS 909
FACTORS INFLUENCING THE
EFFICACY OF MEDIATOR-SPECIFIC
ANTI-INFLAMMATORY,
GLUCOCORTICOID, AND
ANTICOAGULANT THERAPIES
FOR SEPSIS 937
COMBINATORIAL CHEMISTRY IN
THE DRUG DISCOVERY PROCESS 961
HERBAL MEDICINES AND
ANIMAL MODELS OF
GASTROINTESTINAL DISEASES 1013
ENDOCRINE AND
METABOLIC AGENTS 1037
STRATEGIES IN THE DESIGN OF
ANTIVIRAL DRUGS 1135
PROTEIN KINASE INHIBITORS IN
DRUG DISCOVERY 1191
NOVEL IMAGING AGENTS FOR
MOLECULAR MR IMAGING
OF CANCER 1309
TARGETS AND APPROACHES FOR
CANCER DRUG DISCOVERY 1343
MODELING AND INFORMATICS IN
DRUG DESIGN 1375
COMPUTER TECHNIQUES:
IDENTIFYING SIMILARITIES
BETWEEN SMALL MOLECULES 1421
PROTEIN – PROTEIN INTERACTIONS 1461