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 药物发现,开发和制造 499条(本栏目收费,不能显示细节,电话13136136841)
METHOD DEVELOPMENT FOR PRECLINICAL BIOANALYTICAL SUPPORT 1491 
ANALYTICAL CHEMISTRY METHODS: DEVELOPMENTS AND VALIDATION 1525 
CHEMICAL AND PHYSICAL CHARACTERIZATIONS OF POTENTIAL NEW CHEMICAL ENTITY 1585 
PERMEABILITY ASSESSMENT 1601 
HOW AND WHERE ARE DRUGS ABSORBED? 1623 
ABSORPTION OF DRUGS AFTER ORAL ADMINISTRATION 1655 
DISTRIBUTION: MOVEMENT OF DRUGS THROUGH THE BODY 1697 
THE BLOOD – BRAIN BARRIER AND ITS EFFECT ON ABSORPTION AND DISTRIBUTION 1727 
TRANSPORTER INTERACTIONS IN THE ADME PATHWAY OF DRUGS 1781 
ACCUMULATION OF DRUGS IN TISSUES 1803 
SALT AND COCRYSTAL FORM SELECTION 1829 
DISSOLUTION 1857 
STABILITY: PHYSICAL AND CHEMICAL 1919 
DOSAGE FORMULATION 1945 
CYTOCHROME P450 ENZYMES 2001 
METABOLISM KINETICS 2071 
DRUG CLEARANCE 2089 
IN VITRO METABOLISM IN PRECLINICAL DRUG DEVELOPMENT 2117 
UTILIZATION OF IN VITRO CYTOCHROME P450 INHIBITION DATA FOR PROJECTING CLINICAL DRUG – DRUG INTERACTIONS 2149 
IN VIVO METABOLISM IN PRECLINICAL DRUG DEVELOPMENT 2203 
IN VITRO EVALUATION OF METABOLIC DRUG – DRUG INTERACTIONS: SCIENTIFIC CONCEPTS AND PRACTICAL CONSIDERATIONS 2227 
MECHANISMS AND CONSEQUENCES OF DRUG – DRUG INTERACTIONS 2253 
SPECIES COMPARISON OF METABOLISM IN MICROSOMES AND HEPATOCYTES 2293 
METABOLITE PROFILING AND STRUCTURAL IDENTIFICATION 2311 
LINKAGE BETWEEN TOXICOLOGY OF DRUGS AND METABOLISM 2349 
ALLOMETRIC SCALING 2383 
INTERRELATIONSHIP BETWEEN PHARMACOKINETICS AND METABOLISM 2411 
EXPERIMENTAL DESIGN CONSIDERATIONS IN PHARMACOKINETIC STUDIES 2433 
BIOAVAILABILITY AND BIOEQUIVALENCE STUDIES 2443 
MASS BALANCE STUDIES 2477 
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