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靶点信息22(本栏目收费,不能显示细节,电话13136136841)
靶点信息
TARGNAME
Gastric inhibitory polypeptide receptor (GIPR)
TARGTYPE
Clinical trial target
SYNONYMS
Glucosedependent insulinotropic polypeptide receptor; GIPR
FUNCTION
This is a receptor for GIP. The activity of this receptor is mediated by G proteins which activate adenylyl cyclase.
PDBSTRUC
6DKJ; 4HJ0; 2QKH
SEQUENCE
MTTSPILQLLLRLSLCGLLLQRAETGSKGQTAGELYQRWERYRRECQETLAAAEPPSGLACNGSFDMYVCWDYAAPNATARASCPWYLPWHHHVAAGFVLRQCGSDGQWGLWRDHTQCENPEKNEAFLDQRLILERLQVMYTVGYSLSLATLLLALLILSLFRRLHCTRNYIHINLFTSFMLRAAAILSRDRLLPRPGPYLGDQALALWNQALAACRTAQIVTQYCVGANYTWLLVEGVYLHSLLVLVGGSEEGHFRYYLLLGWGAPALFVIPWVIVRYLYENTQCWERNEVKAIWWIIRTPILMTILINFLIFIRILGILLSKLRTRQMRCRDYRLRLARSTLTLVPLLGVHEVVFAPVTEEQARGALRFAKLGFEIFLSSFQGFLVSVLYCFINKEVQSEIRRGWHHCRLRRSLGEEQRQLPERAFRALPSGSGPGEVPTSRGLSSGTLPGPGNEASRELESYC
KEGGPATH
hsa04024:cAMP signaling pathway
KEGGPATH
hsa04080:Neuroactive ligand-receptor interaction
WIKIPATH
WP1824:GPCR downstream signaling
WIKIPATH
WP1825:GPCR ligand binding
WIKIPATH
WP334:GPCRs, Class B Secretin-like
目标的蛋白质ID
标题 | 内容 |
TARGETID |
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UNIPROID |
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TARGNAME |
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TARGTYPE |
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目标的序列数据
标题 | 内容 |
Gastric inhibitory polypeptide receptor (GIPR) |
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