药物发现中的杂环化学 4980条(本栏目收费,不能显示细节,电话13136136841)
2-substituted pyrimidine, 580 580
2-substituted pyrimidine-5-carboxylic esters, 0
synthesis of, 574-575 575
2-substituted quinazolines, amidine in 0
2-substituted quinazolinone, 625 625
synthesis of, 635-636 636
2-substituted thiazoles, 295 295
2-thiosubstituted imidazoles, 343 343
Tykerb (Tyverb), 16, 123-124, 616, 617 617
Type-2 diabetes treatment, 86, 308-309, 359 359
Tyrosine kinase inhibitors (TKIs), 16, 402, 416, 16, 402, 416,
Tyrosine kinase inhibition, 598 598
antihistamine drug for, 311 311
Ulcer treatment, 288, 403 403
Ullmann reaction, in nolatrexed synthesis, 640 640
Ullmann-type coupling, quinazoline derivatives 0
prepared via, 634—635 634—635
Ullmann-type reaction, in imatinib synthesis, 595
Ultrasound irradiation, 443 443
Umpoulong chemistry, 298 298
United States, Imitrex sales in, 56-57 57
Unnatural amino acids, pyridine-containing, 0
Unsaturated amide, 548 548
ct,ß-Unsaturated carbonyl derivatives, amidine 0
Unsaturated ketoximes, 449 449