靶点信息110(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T79961
FORMERID
TTDI01755
UNIPROID
ACM5_HUMAN
TARGNAME
Muscarinic acetylcholine receptor M5 (CHRM5)
GENENAME
CHRM5
TARGTYPE
Successful target
SYNONYMS
CHRM5
FUNCTION
After binding acetylcholine, the AChR responds by an extensive change in conformation that affects all subunits and leads to opening of an ion-conducting channel across the plasma membrane.
BIOCLASS
GPCR rhodopsin
SEQUENCE
MEGDSYHNATTVNGTPVNHQPLERHRLWEVITIAAVTAVVSLITIVGNVLVMISFKVNSQLKTVNNYYLLSLACADLIIGIFSMNLYTTYILMGRWALGSLACDLWLALDYVASNASVMNLLVISFDRYFSITRPLTYRAKRTPKRAGIMIGLAWLISFILWAPAILCWQYLVGKRTVPLDECQIQFLSEPTITFGTAIAAFYIPVSVMTILYCRIYRETEKRTKDLADLQGSDSVTKAEKRKPAHRALFRSCLRCPRPTLAQRERNQASWSSSRRSTSTTGKPSQATGPSANWAKAEQLTTCSSYPSSEDEDKPATDPVLQVVYKSQGKESPGEEFSAEETEETFVKAETEKSDYDTPNYLLSPAAAHRPKSQKCVAYKFRLVVKADGNQETNNGCHKVKIMPCPFPVAKEPSTKGLNPNPSHQMTKRKRVVLVKERKAAQTLSAILLAFIITWTPYNIMVLVSTFCDKCVPVTLWHLGYWLCYVNSTVNPICYALCNRTFRKTFKMLLLCRWKKKKVEEKLYWQGNSKLP
DRUGINFO
ACECLIDINE
DRUGINFO
Anisodine
DRUGINFO
Anisotropine Methylbromide
DRUGINFO
Atropine
DRUGINFO
Belladonna
DRUGINFO
Bethanechol
DRUGINFO
Butylscopolamine
DRUGINFO
Choline alfoscerate
DRUGINFO
Cimetropium bromide
DRUGINFO
Cryptenamine Acetates
目标的 KEGG 通路数据
标题内容
hsa04020
hsa04080
hsa04725
hsa04810
目标的 Wiki 路径数据
标题内容
WP58
WP536
WP51
WP455
WP2664
WP1825
WP1824
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
Muscarinic acetylcholine receptor M5 (CHRM5)
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