靶点信息43(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T78581
FORMERID
TTDR00184
UNIPROID
GALR1_HUMAN
TARGNAME
Galanin receptor type 1 (GAL1-R)
GENENAME
GALR1
TARGTYPE
Literature-reported target
SYNONYMS
GALR1; GALR-1; GALNR1; GALN1R; GAL1-R
FUNCTION
The activity of this receptor is mediated by G proteins that inhibit adenylate cyclase activity. Receptor for the hormone galanin. G protein-coupled peptide receptor activity. Neuropeptide binding. Peptide hormone binding.
BIOCLASS
GPCR rhodopsin
SEQUENCE
MELAVGNLSEGNASWPEPPAPEPGPLFGIGVENFVTLVVFGLIFALGVLGNSLVITVLARSKPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLVSIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGCIWALSIAMASPVAYHQGLFHPRASNQTFCWEQWPDPRHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASKKKTAQTVLVVVVVFGISWLPHHIIHLWAEFGVFPLTPASFLFRITAHCLAYSNSSVNPIIYAFLSENFRKAYKQVFKCHIRKDSHLSDTKESKSRIDTPPSTNCTHV
DRUGINFO
(Sar)WTLNSAGYLLGPKK(Lys-decanoyl)K
DRUGINFO
(Sar)WTLNSAGYLLGPKK(Lys-lauroyl)K
DRUGINFO
(Sar)WTLNSAGYLLGPKK(Lys-MPEG4)K
DRUGINFO
(Sar)WTLNSAGYLLGPKK(Lys-myristoyl)K
DRUGINFO
(Sar)WTLNSAGYLLGPKK(Lys-octanoyl)K
DRUGINFO
(Sar)WTLNSAGYLLGPKK(Lys-palmitoyl)K
DRUGINFO
(Sar)WTLNSAGYLLGPKK(Lys-stearoyl)K
DRUGINFO
(Sar)WTLNSAGYLLGPKKKK
DRUGINFO
[N-Ac,des-Sar]Gal-B2
DRUGINFO
[N-Me,des-Sar]Gal-B2
目标的 KEGG 通路数据
标题内容
hsa04080
目标的 Wiki 路径数据
标题内容
WP455
WP24
WP1825
WP1824
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
Galanin receptor type 1 (GAL1-R)
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