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靶点信息82(本栏目收费,不能显示细节,电话13136136841)
靶点信息
TARGNAME
Thromboxane A2 receptor (TBXA2R)
TARGTYPE
Successful target
SYNONYMS
TXA2-R; TXA2 receptor; Prostanoid TP receptor
FUNCTION
The activity of this receptor is mediated by a G-protein that activates a phosphatidylinositol-calcium second messenger system. In the kidney, the binding of TXA2 to glomerular TP receptors causes intense vasoconstriction. Activates phospholipase C. Isoform 1 activates adenylyl cyclase. Isoform 2 inhibits adenylyl cyclase. Receptor for thromboxane A2 (TXA2), a potent stimulator of platelet aggregation.
SEQUENCE
MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTRSSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPLLLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPGSWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSEVEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWNQILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
DRUGINFO
Ifetroban sodium
目标的 KEGG 通路数据
标题 | 内容 |
hsa04020 |
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hsa04080 |
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hsa04611 |
|
目标的 Wiki 路径数据
标题 | 内容 |
WP455 |
|
WP2664 |
|
WP247 |
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WP1908 |
|
WP1825 |
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WP1824 |
|
目标的蛋白质ID
标题 | 内容 |
TARGETID |
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UNIPROID |
|
TARGNAME |
|
TARGTYPE |
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目标的序列数据
标题 | 内容 |
Thromboxane A2 receptor (TBXA2R) |
|