靶点信息27(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T22032
FORMERID
TTDC00041
UNIPROID
PTH2R_HUMAN
TARGNAME
Parathyroid hormone receptor (PTH2R)
GENENAME
PTH2R
TARGTYPE
Clinical trial target
SYNONYMS
PTHR2; PTH2R; PTH2 receptor
FUNCTION
This is a specific receptor for parathyroid hormone. The activity of this receptor is mediated by G proteins which activate adenylyl cyclase. PTH2R may be responsible for PTH effects in a number of physiological systems. It may play asignificant role in pancreatic function. PTH2R presence in neurons indicates that it may function as a neurotransmitter receptor.
BIOCLASS
GPCR secretin
SEQUENCE
MAGLGASLHVWGWLMLGSCLLARAQLDSDGTITIEEQIVLVLKAKVQCELNITAQLQEGEGNCFPEWDGLICWPRGTVGKISAVPCPPYIYDFNHKGVAFRHCNPNGTWDFMHSLNKTWANYSDCLRFLQPDISIGKQEFFERLYVMYTVGYSISFGSLAVAILIIGYFRRLHCTRNYIHMHLFVSFMLRATSIFVKDRVVHAHIGVKELESLIMQDDPQNSIEATSVDKSQYIGCKIAVVMFIYFLATNYYWILVEGLYLHNLIFVAFFSDTKYLWGFILIGWGFPAAFVAAWAVARATLADARCWELSAGDIKWIYQAPILAAIGLNFILFLNTVRVLATKIWETNAVGHDTRKQYRKLAKSTLVLVLVFGVHYIVFVCLPHSFTGLGWEIRMHCELFFNSFQGFFVSIIYCYCNGEVQAEVKKMWSRWNLSVDWKRTPPCGSRRCGSVLTTVTHSTSSQSQVAASTRMVLISGKAAKIASRQPDSHITLPGYVWSNSEQDCLPHSFHEETKEDSGRQGDDILMEKPSRPMESNPDTEGCQGETEDVL
DRUGINFO
BA-058
DRUGINFO
GSK768974
DRUGINFO
NPSP-795
DRUGINFO
UNI-PH (1-34)
DRUGINFO
PTH(7-34) liposomal cream
DRUGINFO
Semparatide
DRUGINFO
BB-PTH 1-84
DRUGINFO
Hemoparatide
DRUGINFO
PTHr pepducins
DRUGINFO
SDZ-PTS-893
目标的 KEGG 通路数据
标题内容
hsa04080
目标的 Wiki 路径数据
标题内容
WP334
WP1825
WP1824
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
Parathyroid hormone receptor (PTH2R)
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