靶点信息19(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T21865
FORMERID
TTDR01112
UNIPROID
SELPL_HUMAN
TARGNAME
P-selectin glycoprotein ligand 1 (SELPLG)
GENENAME
SELPLG
TARGTYPE
Clinical trial target
SYNONYMS
Selectin P ligand; SPSGL-1; SELPLG; PSGL-1; P-selectin glycoprotein ligand-1; CD162 antigen
FUNCTION
A SLe(x)-type proteoglycan, which through high affinity, calcium-dependent interactions with E-, P- and L-selectins, mediates rapid rolling of leukocytes over vascular surfaces during the initial steps in inflammation. Critical for the initial leukocyte capture.
PDBSTRUC
1G1S
SEQUENCE
MPLQLLLLLILLGPGNSLQLWDTWADEAEKALGPLLARDRRQATEYEYLDYDFLPETEPPEMLRNSTDTTPLTGPGTPESTTVEPAARRSTGLDAGGAVTELTTELANMGNLSTDSAAMEIQTTQPAATEAQTTQPVPTEAQTTPLAATEAQTTRLTATEAQTTPLAATEAQTTPPAATEAQTTQPTGLEAQTTAPAAMEAQTTAPAAMEAQTTPPAAMEAQTTQTTAMEAQTTAPEATEAQTTQPTATEAQTTPLAAMEALSTEPSATEALSMEPTTKRGLFIPFSVSSVTHKGIPMAASNLSVNYPVGAPDHISVKQCLLAILILALVATIFFVCTVVLAVRLSRKGHMYPVRNYSPTEMVCISSLLPDGGEGPSATANGGLSKAKSPGLTPEPREDREGDDLTLHSFLP
DRUGINFO
AbGn-168
DRUGINFO
Neihulizumab
DRUGINFO
RO-4905417
KEGGPATH
hsa04514:Cell adhesion molecules (CAMs)
KEGGPATH
hsa05150:Staphylococcus aureus infection
WIKIPATH
WP1794:Cell surface interactions at the vascular wall
WIKIPATH
WP2806:Human Complement System
REACPATH
R-HSA-202733:Cell surface interactions at the vascular wall
INTEPATH
amb2_neutrophils_pathway:amb2 Integrin signaling
目标的 KEGG 通路数据
标题内容
hsa04514
hsa05150
目标的 Wiki 路径数据
标题内容
WP2806
WP1794
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
P-selectin glycoprotein ligand 1 (SELPLG)
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