靶点信息27(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T20575
FORMERID
TTDR00763
UNIPROID
CCR8_HUMAN
TARGNAME
C-C chemokine receptor type 8 (CCR8)
GENENAME
CCR8
TARGTYPE
Discontinued target
SYNONYMS
TER1; GPRCY6; GPR-CY6; Chemokine receptor-like 1; Chemokine receptor CCR8; CMKBRL2; CMKBR8; CKRL1; CKR-L1; CDw198; CCR-8; CC-chemokine receptor CHEMR1; CC-CKR-8; CC chemokine receptor CHEMR1; C-C CKR-8
FUNCTION
May regulate monocyte chemotaxis and thymic cell line apoptosis. Alternative coreceptor with CD4 for HIV-1 infection. Receptor for the chemokine CCL1/SCYA1/I-309.
BIOCLASS
GPCR rhodopsin
SEQUENCE
MDYTLDLSVTTVTDYYYPDIFSSPCDAELIQTNGKLLLAVFYCLLFVFSLLGNSLVILVLVVCKKLRSITDVYLLNLALSDLLFVFSFPFQTYYLLDQWVFGTVMCKVVSGFYYIGFYSSMFFITLMSVDRYLAVVHAVYALKVRTIRMGTTLCLAVWLTAIMATIPLLVFYQVASEDGVLQCYSFYNQQTLKWKIFTNFKMNILGLLIPFTIFMFCYIKILHQLKRCQNHNKTKAIRLVLIVVIASLLFWVPFNVVLFLTSLHSMHILDGCSISQQLTYATHVTEIISFTHCCVNPVIYAFVGEKFKKHLSEIFQKSCSQIFNYLGRQMPRESCEKSSSCQQHSSRSSSVDYIL
DRUGINFO
I-309
DRUGINFO
N-(4-phenylsulfamoyl-naphthalen-1-yl)-benzamide
DRUGINFO
N-{4-[(benzylamino)sulfonyl]-1-naphthyl}benzamide
DRUGINFO
viral macrophage inflammatory protein-II
DRUGINFO
ZK 756326
KEGGPATH
hsa04060:Cytokine-cytokine receptor interaction
KEGGPATH
hsa04062:Chemokine signaling pathway
KEGGPATH
hsa05203:Viral carcinogenesis
WIKIPATH
WP1824:GPCR downstream signaling
目标的 KEGG 通路数据
标题内容
hsa04060
hsa04062
hsa05203
目标的 Wiki 路径数据
标题内容
WP455
WP24
WP1825
WP1824
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
C-C chemokine receptor type 8 (CCR8)
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