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靶点信息67(本栏目收费,不能显示细节,电话13136136841)
靶点信息
TARGNAME
Somatostatin receptor type 1 (SSTR1)
TARGTYPE
Successful target
SYNONYMS
Sst(1); Somatostatin receptor 1; SSTR1; SS1R; SRIF-2
FUNCTION
Receptor for somatostatin with higher affinity for somatostatin-14 than -28. This receptor is coupled via pertussis toxin sensitive G proteins to inhibition of adenylyl cyclase. In addition it stimulates phosphotyrosine phosphataseand Na(+)/H(+) exchanger via pertussis toxin insensitive G proteins.
SEQUENCE
MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAILISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLLRHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLGVWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAICLCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQDDATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKSRAYSVEDFQPENLESGGVFRNGTCTSRITTL
DRUGINFO
Lutetium Lu 177 dotatate
DRUGINFO
Cytotoxin Peptide Conjugate
DRUGINFO
Des-AA1,2,4,12,13-[D-Trp8]SRIF
DRUGINFO
Des-AA1,2,4,13-[D-Trp8]SRIF
DRUGINFO
Des-AA1,2,4,5,13-[D-Trp8]-SRIF
目标的 Wiki 路径数据
标题 | 内容 |
WP706 |
|
WP455 |
|
WP24 |
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WP1825 |
|
WP1824 |
|
目标的蛋白质ID
标题 | 内容 |
TARGETID |
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UNIPROID |
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TARGNAME |
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TARGTYPE |
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目标的序列数据
标题 | 内容 |
Somatostatin receptor type 1 (SSTR1) |
|