靶点信息105(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T11448
FORMERID
TTDS00032
UNIPROID
ADA2A_HUMAN
TARGNAME
Adrenergic receptor alpha-2A (ADRA2A)
GENENAME
ADRA2A
TARGTYPE
Successful target
SYNONYMS
Alpha-2AAR; Alpha-2A adrenoreceptor; Alpha-2A adrenoceptor; Alpha-2A adrenergic receptor; Alpha-2 adrenergic receptor subtype C10; ADRAR; ADRA2R
FUNCTION
The rank order of potency for agonists of this receptor is oxymetazoline > clonidine > epinephrine > norepinephrine > phenylephrine > dopamine > p-synephrine > p-tyramine > serotonin = p-octopamine. For antagonists, the rank order is yohimbine > phentolamine = mianserine > chlorpromazine = spiperone = prazosin > propanolol > alprenolol = pindolol. Alpha-2 adrenergic receptors mediate the catecholamine-induced inhibition of adenylate cyclase through the action of G proteins.
PDBSTRUC
1HOF; 1HOD; 1HO9; 1HLL
BIOCLASS
GPCR rhodopsin
SEQUENCE
MFRQEQPLAEGSFAPMGSLQPDAGNASWNGTEAPGGGARATPYSLQVTLTLVCLAGLLMLLTVFGNVLVIIAVFTSRALKAPQNLFLVSLASADILVATLVIPFSLANEVMGYWYFGKAWCEIYLALDVLFCTSSIVHLCAISLDRYWSITQAIEYNLKRTPRRIKAIIITVWVISAVISFPPLISIEKKGGGGGPQPAEPRCEINDQKWYVISSCIGSFFAPCLIMILVYVRIYQIAKRRTRVPPSRRGPDAVAAPPGGTERRPNGLGPERSAGPGGAEAEPLPTQLNGAPGEPAPAGPRDTDALDLEESSSSDHAERPPGPRRPERGPRGKGKARASQVKPGDSLPRRGPGATGIGTPAAGPGEERVGAAKASRWRGRQNREKRFTFVLAVVIGVFVVCWFPFFFTYTLTAVGCSVPRTLFKFFFWFGYCNSSLNPVIYTIFNHDFRRAFKKILCRGDRKRIV
DRUGINFO
Connexyn
DRUGINFO
Lofexidine
DRUGINFO
MOXONIDINE
DRUGINFO
MEDETOMIDINE
DRUGINFO
DSP-1200
DRUGINFO
MAZAPERTINE
DRUGINFO
A-80426
DRUGINFO
S-18616
目标的 KEGG 通路数据
标题内容
hsa04022
hsa04080
目标的 Wiki 路径数据
标题内容
WP58
WP455
WP1884
WP1831
WP1825
WP1824
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
Adrenergic receptor alpha-2A (ADRA2A)
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