靶点信息63(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T11241
FORMERID
TTDI02523
UNIPROID
S1PR3_HUMAN
TARGNAME
Sphingosine-1-phosphate receptor 3 (S1PR3)
GENENAME
S1PR3
TARGTYPE
Patented-recorded target
SYNONYMS
Sphingosine 1-phosphate receptor Edg-3; S1PR3; S1P3; S1P receptor Edg-3; S1P receptor 3; Endothelial differentiation G-protein coupled receptor 3
FUNCTION
Receptor for the lysosphingolipid sphingosine 1- phosphate (S1P). S1P is a bioactive lysophospholipid that elicits diverse physiological effect on most types of cells and tissues. When expressed in rat HTC4 hepatoma cells, is capable of mediating S1P-induced cell proliferation and suppression of apoptosis.
BIOCLASS
GPCR rhodopsin
SEQUENCE
MATALPPRLQPVRGNETLREHYQYVGKLAGRLKEASEGSTLTTVLFLVICSFIVLENLMVLIAIWKNNKFHNRMYFFIGNLALCDLLAGIAYKVNILMSGKKTFSLSPTVWFLREGSMFVALGASTCSLLAIAIERHLTMIKMRPYDANKRHRVFLLIGMCWLIAFTLGALPILGWNCLHNLPDCSTILPLYSKKYIAFCISIFTAILVTIVILYARIYFLVKSSSRKVANHNNSERSMALLRTVVIVVSVFIACWSPLFILFLIDVACRVQACPILFKAQWFIVLAVLNSAMNPVIYTLASKEMRRAFFRLVCNCLVRGRGARASPIQPALDPSRSKSSSSNNSSHSPKVKEDLPHTAPSSCIMDKNAALQNGIFCN
DRUGINFO
BDBM50080559
DRUGINFO
BDBM50080563
DRUGINFO
BDBM50080570
DRUGINFO
JCXGHZCWAHCYGY-UHFFFAOYSA-N
DRUGINFO
MHHFJYABEVJNEG-UHFFFAOYSA-N
DRUGINFO
US10166249, Example 695
DRUGINFO
US10179791, Compound 171
DRUGINFO
US10179791, Compound 176
DRUGINFO
US10179791, Compound 296
DRUGINFO
US8524917, 10
目标的 KEGG 通路数据
标题内容
hsa04071
hsa04080
目标的 Wiki 路径数据
标题内容
WP26
WP247
WP1825
WP1824
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
Sphingosine-1-phosphate receptor 3 (S1PR3)
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