靶点信息37(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T10091
FORMERID
TTDR00221
UNIPROID
OPSD_HUMAN
TARGNAME
Rhodopsin (RHO)
GENENAME
RHO
TARGTYPE
Literature-reported target
SYNONYMS
Opsin-2; OPN2
FUNCTION
Required for photoreceptor cell viability after birth. Light-induced isomerization of the chromophore 11-cis-retinal to all-trans-retinal triggers a conformational change that activates signaling via G-proteins. Subsequent receptor phosphorylation mediates displacement of the bound G-protein alpha subunit by the arrestin SAG and terminates signaling. Photoreceptor required for image-forming vision at low light intensity.
PDBSTRUC
6CMO; 5W0P; 5DGY; 4ZWJ
BIOCLASS
GPCR rhodopsin
SEQUENCE
MNGTEGPNFYVPFSNATGVVRSPFEYPQYYLAEPWQFSMLAAYMFLLIVLGFPINFLTLYVTVQHKKLRTPLNYILLNLAVADLFMVLGGFTSTLYTSLHGYFVFGPTGCNLEGFFATLGGEIALWSLVVLAIERYVVVCKPMSNFRFGENHAIMGVAFTWVMALACAAPPLAGWSRYIPEGLQCSCGIDYYTLKPEVNNESFVIYMFVVHFTIPMIIIFFCYGQLVFTVKEAAAQQQESATTQKAEKEVTRMVIIMVIAFLICWVPYASVAFYIFTHQGSNFGPIFMTIPAFFAKSAAIYNPVIYIMMNKQFRNCMLTTICCGKNPLGDDEASATVSKTETSQVAPA
DRUGINFO
(Hydroxyethyloxy)Tri(Ethyloxy)Octane
DRUGINFO
Alpha-D-Mannose
DRUGINFO
B-2-Octylglucoside
DRUGINFO
Beta-D-Mannose
DRUGINFO
B-Nonylglucoside
DRUGINFO
B-Octylglucoside
DRUGINFO
Heptane-1,2,3-Triol
DRUGINFO
Heptyl 1-Thiohexopyranoside
DRUGINFO
Hexadecanal
目标的 KEGG 通路数据
标题内容
hsa04744
目标的 Wiki 路径数据
标题内容
WP455
WP2776
WP2038
WP1984
WP185
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
Rhodopsin (RHO)
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