靶点信息62(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T09960
FORMERID
TTDS00326
UNIPROID
CCR5_HUMAN
TARGNAME
C-C chemokine receptor type 5 (CCR5)
GENENAME
CCR5
TARGTYPE
Successful target
SYNONYMS
HIV-1 fusion coreceptor; HIV-1 fusion co-receptor; Chemokine receptor CCR5; CMKBR5; CHEMR13; CD195 antigen; CD195; CCR-5; CC-CKR-5; C-C CKR-5
FUNCTION
May play a role in the control of granulocytic lineage proliferation or differentiation. Receptor for a number of inflammatory CC-chemokines including CCL3/MIP-1-alpha, CCL4/MIP-1-beta and RANTES and subsequently transduces a signal by increasing the intracellular calcium ion level.
PDBSTRUC
6MET; 6MEO; 6FGP; 5YY4; 5YD5
BIOCLASS
GPCR rhodopsin
SEQUENCE
MDYQVSSPIYDINYYTSEPCQKINVKQIAARLLPPLYSLVFIFGFVGNMLVILILINCKRLKSMTDIYLLNLAISDLFFLLTVPFWAHYAAAQWDFGNTMCQLLTGLYFIGFFSGIFFIILLTIDRYLAVVHAVFALKARTVTFGVVTSVITWVVAVFASLPGIIFTRSQKEGLHYTCSSHFPYSQYQFWKNFQTLKIVILGLVLPLLVMVICYSGILKTLLRCRNEKKRHRAVRLIFTIMIVYFLFWAPYNIVLLLNTFQEFFGLNNCSSSNRLDQAMQVTETLGMTHCCINPIIYAFVGEKFRNYLLVFFQKHIAKRFCKCCSIFQQEAPERASSVYTRSTGEQEISVGL
DRUGINFO
Maraviroc
DRUGINFO
E-913
DRUGINFO
PRO-140
DRUGINFO
Vicriviroc
DRUGINFO
PRO 140
DRUGINFO
INCB9471
DRUGINFO
BMS-813160
DRUGINFO
Cenicriviroc
DRUGINFO
GSK-706769
目标的 KEGG 通路数据
标题内容
hsa04060
hsa04062
hsa04144
hsa05145
hsa05203
目标的 Wiki 路径数据
标题内容
WP69
WP455
WP2658
WP24
WP1825
WP1824
WP117
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
C-C chemokine receptor type 5 (CCR5)
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