靶点信息74(本栏目收费,不能显示细节,电话13136136841)
靶点信息
标题
内容
相关药物
状态
TARGETID
T02001
FORMERID
TTDS00499
UNIPROID
PDE4D_HUMAN
TARGNAME
Phosphodiesterase 4D (PDE4D)
GENENAME
PDE4D
TARGTYPE
Successful target
SYNONYMS
cAMP-specific 3',5'-cyclic phosphodiesterase 4D; PDE43; DPDE3
FUNCTION
Hydrolyzes the second messenger cAMP, which is a key regulator of many important physiological processes.
PDBSTRUC
6NJJ; 6NJI; 6NJH; 6FW3; 6FTW
BIOCLASS
Phosphoric diester hydrolase
ECNUMBER
EC 3.1.4.53
SEQUENCE
MEAEGSSAPARAGSGEGSDSAGGATLKAPKHLWRHEQHHQYPLRQPQFRLLHPHHHLPPPPPPSPQPQPQCPLQPPPPPPLPPPPPPPGAARGRYASSGATGRVRHRGYSDTERYLYCRAMDRTSYAVETGHRPGLKKSRMSWPSSFQGLRRFDVDNGTSAGRSPLDPMTSPGSGLILQANFVHSQRRESFLYRSDSDYDLSPKSMSRNSSIASDIHGDDLIVTPFAQVLASLRTVRNNFAALTNLQDRAPSKRSPMCNQPSINKATITEEAYQKLASETLEELDWCLDQLETLQTRHSVSEMASNKFKRMLNRELTHLSEMSRSGNQVSEFISNTFLDKQHEVEIPSPTQKEKEKKKRPMSQISGVKKLMHSSSLTNSSIPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQSPSPAPDDPEEGRQGQTEKFQFELTLEEDGESDTEKDSGSQVEEDTSCSDSKTLCTQDSESTEIPLDEQVEEEAVGEEEESQPEACVIDDRSPDT
DRUGINFO
Papaverine
DRUGINFO
DENBUFYLLINE
DRUGINFO
SOTB07
DRUGINFO
AN-2898
DRUGINFO
AWD-12-281
DRUGINFO
BPN14770
DRUGINFO
CC-1088
DRUGINFO
GPD-1116
目标的 KEGG 通路数据
标题内容
hsa00230
hsa04024
hsa05032
目标的 Wiki 路径数据
标题内容
WP35
WP289
WP2032
目标的蛋白质ID
标题内容
TARGETID
UNIPROID
TARGNAME
TARGTYPE
目标的序列数据
标题内容
Phosphodiesterase 4D (PDE4D)
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