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靶点信息47(本栏目收费,不能显示细节,电话13136136841)
靶点信息
TARGNAME
Neuropeptide Y receptor type 1 (NPY1R)
TARGTYPE
Clinical trial target
SYNONYMS
Neuropeptide Y-Y1 receptor; Neuropeptide Y receptor Y1; Neuropeptide Y Y(1) receptor; NPY1R; NPY1-R
FUNCTION
Receptor for neuropeptide Y and peptide YY. The rank order of affinity of this receptor for pancreatic polypeptides is NPY > [Pro-34] PYY, PYY and [Leu-31, Pro-34] NPY > NPY (2-36) > [Ile-31, Gln-34] PP and PYY (3-36) > PP > NPY free acid.
PDBSTRUC
5ZBQ; 2IIL; 2F1U
SEQUENCE
MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMTDEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKINNNDDNEKI
DRUGINFO
[Cys-Trp-Arg-Nva-Arg-Tyr-NH2]2
DRUGINFO
4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one
目标的 Wiki 路径数据
标题 | 内容 |
WP455 |
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WP24 |
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WP2197 |
|
WP1825 |
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WP1824 |
|
目标的蛋白质ID
标题 | 内容 |
TARGETID |
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UNIPROID |
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TARGNAME |
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TARGTYPE |
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目标的序列数据
标题 | 内容 |
Neuropeptide Y receptor type 1 (NPY1R) |
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