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靶点信息65(本栏目收费,不能显示细节,电话13136136841)
靶点信息
TARGNAME
Melanocortin receptor 3 (MC3R)
TARGTYPE
Literature-reported target
FUNCTION
Receptor for MSH (alpha, beta and gamma) and ACTH. This receptor is mediated by G proteins which activate adenylate cyclase. Required for expression of anticipatory patterns of activity and wakefulness during periods of limited nutrient availability and for the normal regulation of circadian clock activity in the brain.
SEQUENCE
MNASCCLPSVQPTLPNGSEHLQAPFFSNQSSSAFCEQVFIKPEVFLSLGIVSLLENILVILAVVRNGNLHSPMYFFLCSLAVADMLVSVSNALETIMIAIVHSDYLTFEDQFIQHMDNIFDSMICISLVASICNLLAIAVDRYVTIFYALRYHSIMTVRKALTLIVAIWVCCGVCGVVFIVYSESKMVIVCLITMFFAMMLLMGTLYVHMFLFARLHVKRIAALPPADGVAPQQHSCMKGAVTITILLGVFIFCWAPFFLHLVLIITCPTNPYCICYTAHFNTYLVLIMCNSVIDPLIYAFRSLELRNTFREILCGCNGMNLG
DRUGINFO
Ac-[CEHdFRWC]-NH2
DRUGINFO
Ac-dR[CEHdFRWC]-NH2
DRUGINFO
Ac-His-D-Phe-Arg-2-Nal-NHCH3
DRUGINFO
Ac-Nle-c[Asp-His-DNal(2')-Pro-Trp-Lys]-NH2
DRUGINFO
Ac-R[CEHdFRWC]-NH2
DRUGINFO
Ac-Tyr-D-Phe-Arg-2-Nal-NHCH3
DRUGINFO
Ac-YCit[CEHdFRWC]-NH2
DRUGINFO
Ac-YK[CEHdFRWC]-NH2
DRUGINFO
Ac-YR[CEH(d-2alpha-Nal)RWC]-NH2
目标的 Wiki 路径数据
标题 | 内容 |
WP455 |
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WP24 |
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WP1825 |
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WP1824 |
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目标的蛋白质ID
标题 | 内容 |
TARGETID |
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UNIPROID |
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TARGNAME |
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TARGTYPE |
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目标的序列数据
标题 | 内容 |
Melanocortin receptor 3 (MC3R) |
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