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靶点信息61(本栏目收费,不能显示细节,电话13136136841)
靶点信息
TARGNAME
Orexin receptor type 2 (HCRTR2)
TARGTYPE
Successful target
SYNONYMS
Ox2r; Ox2-R; Ox-2-R; Orexin-2 receptor; Hypocretin receptor type 2; HFGANP
FUNCTION
Triggers an increase in cytoplasmic Ca(2+) levels in response to orexin-A binding. Nonselective, high-affinity receptor for both orexin-A and orexin-B neuropeptides.
PDBSTRUC
5WS3; 5WQC; 4S0V
SEQUENCE
MSGTKLEDSPPCRNWSSASELNETQEPFLNPTDYDDEEFLRYLWREYLHPKEYEWVLIAGYIIVFVVALIGNVLVCVAVWKNHHMRTVTNYFIVNLSLADVLVTITCLPATLVVDITETWFFGQSLCKVIPYLQTVSVSVSVLTLSCIALDRWYAICHPLMFKSTAKRARNSIVIIWIVSCIIMIPQAIVMECSTVFPGLANKTTLFTVCDERWGGEIYPKMYHICFFLVTYMAPLCLMVLAYLQIFRKLWCRQIPGTSSVVQRKWKPLQPVSQPRGPGQPTKSRMSAVAAEIKQIRARRKTARMLMIVLLVFAICYLPISILNVLKRVFGMFAHTEDRETVYAWFTFSHWLVYANSAANPIIYNFLSGKFREEFKAAFSCCCLGVHHRQEDRLTRGRTSTESRKSLTTQISNFDNISKLSEQVVLTSISTLPAANGAGPLQNW
DRUGINFO
1,2-diamino cyclopentane-based derivative 1
DRUGINFO
1,2-diamino cyclopentane-based derivative 10
DRUGINFO
1,2-diamino cyclopentane-based derivative 11
DRUGINFO
1,2-diamino cyclopentane-based derivative 12
DRUGINFO
1,2-diamino cyclopentane-based derivative 13
DRUGINFO
1,2-diamino cyclopentane-based derivative 14
目标的 Wiki 路径数据
标题 | 内容 |
WP455 |
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WP2664 |
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WP1825 |
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WP1824 |
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目标的蛋白质ID
标题 | 内容 |
TARGETID |
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UNIPROID |
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TARGNAME |
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TARGTYPE |
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目标的序列数据
标题 | 内容 |
Orexin receptor type 2 (HCRTR2) |
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